Ibicuruzwa

Itandukaniro riraboneka

N / a

Ibikoresho

  • Irashobora gufasha kurwanya antimalarial

Artemether cas 71963-77-4 Artemisia Annua Kureka

Artemether CAS 71963-77-4 Artemisia Annua ibikuremo ishusho

Ibisobanuro birambuye

Ibicuruzwa

Itandukaniro N / a
CAS OYA 71963-77-4
Formulaire C16H26O5
Uburemere bwa molekile 298.37
EINIONC no. 663-549-0
Gushonga 86-88 ° C.
Ingingo itetse 359.79 ° C (Ikigereranyo kitoroshye)
Kuzunguruka D19.5 + 171 ° (C = 2.59Inchcl3)
Ubucucike 1.0733 (Ikigereranyo kitoroshye)
Indangagaciro yo gutunganya 1.6200 (Ikigereranyo)
Imiterere Icyumba
Kudashoboka DMSO≥20MG / ML
Isura Ifu
Synonyme Artemetherum / Artemtherin / Ibihe Byahe
Kudashoboka Gushonga mumazi
Ibyiciro Gukuramo ibimera, inyongera, ubuvuzi
Porogaramu Kurwanya malarial

Artemether ni lactiterpene lactine iboneka mumizi yaArtemisia Annua, mubisanzwe bizwi nka Wormwood nziza. Numuti ukaze urwanya ukoreshwa mugufata no kwirinda malariya. Artemisinin, ibanziriza artemether, yakuwe mu gihingwa cya mbere mu myaka ya za 70, kandi kuvumbura kwavumburwa byibuze mu Bushinwa Tu YoUUUre igihembo cyitiriwe mu buti muri 2015.

Artemether ikora mugusenya parasite ishinzwe guteza malariya. Malariya iterwa na parasite ya protozoan yitwa plasmodium, ishyikirizwa abantu binyuze mu kuruma imibu ya anofephitoes zanduye. Amaze kwinjira mu ngabo, parasite kugwira vuba mu mwijima na selile itukura, bigatera umuriro, gukonja, n'ibindi bimenyetso nk'ibicurane. Iyo itavuwe, malariya irashobora kwica.

Artemether ningirakamaro cyane kurwanya imiti irwanya ibiyobyabwenge ya Falcitum ya Plasmodium, niyihe konti yatumye impfu ziterwa na malariya. Ikora kandi kurwanya ubundi bwoko bwa parasite ya plasmodium itera malariya. Ubusanzwe Artemether iyobowe nibiyobyabwenge, nka lumefantrine, kugirango bigabanye ibyago byo kurwanya ibiyobyabwenge.

Usibye gukoresha nk'ibiyobyabwenge byo kurwanya antimalarial, artemether na we wasangaga ufite ubundi buryo bwo kuvura. Ubushakashatsi bwerekanye ko bufite anti-indumu, kurwanya ibibyimba, no kurwanya virusi. Byakoreshejwe mukuvura arthritis, lupus, nizindi ndwara za automune. Yarekuwe kandi ku bushobozi bwaryo bwo gufata Covid - 19, nubwo hakenewe ubushakashatsi bwo kwemeza imikorere yayo.

Artemether muri rusange afite umutekano kandi yihanganiye neza mugihe yakoreshejwe nkuko byateganijwe. Ariko, kimwe nibiyobyabwenge byose, birashobora gutera ingaruka. Ingaruka zisanzwe za ardemest zirimo isesemi, kuruka, kuzunguruka, no kubabara umutwe. Mubibazo bidasanzwe, birashobora gutera ibintu bibi nkibi, nko kurandura umutima, gufatwa, no kwangiza umwijima.

Mu gusoza, Artemether ni ibiyobyabwenge bikomeye bidasanzwe byahinduye imiti no gukumira malariya. Ubuvumbuzi bwayo bwazigamye ubuzima butabarika kandi bwinjije kubaturage ba siyansi. Ibindi byatangaga byumutungo bigira umukandida utanga icyizere kugirango tuvure izindi ndwara. Nubwo bishobora gutera ingaruka, inyungu zayo ziruta kure ingaruka zayo mugihe zikoreshwa mubuvuzi.
Impapuro zikoreshwa zisanzwe zirimo ibisate, capsules no gutera inshinge. Ubwoko bw'ibiyobyabwenge ni ibiyobyabwenge birwanya, kandi ibintu nyamukuru ni artemether. Imiterere yimpamvu ya Artemertert yari ibinini byera. Imiterere ya ardemether capsule ni capsule, ibikubiye muri byo ni ifu yera; Imiterere y'ibiyobyabwenge yo gutera inshinge nta mari yamabara yumuhondo - nkamazi.

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